A Pilot Study of BMS-512148 in Subjects With Type 2 Diabetes

This study has been completed.
Sponsor:
Information provided by:
Bristol-Myers Squibb
ClinicalTrials.gov Identifier:
NCT00357370
First received: July 26, 2006
Last updated: September 10, 2010
Last verified: July 2009
  Purpose

The purpose of this clinical research study is to learn if BMS-512148, added to insulin and one or two anti-diabetes medications (metformin and/or pioglitazone or rosiglitazone), can help reduce the blood sugar levels compared to insulin and one or two anti-diabetes medications (metformin and/or pioglitazone or rosiglitazone) alone, in subjects with type 2 diabetes. The safety of this treatment will also be studied.


Condition Intervention Phase
Type 2 Diabetes
Drug: Dapagliflozin
Drug: Placebo
Phase 2
Phase 3

Study Type: Interventional
Study Design: Allocation: Randomized
Endpoint Classification: Safety/Efficacy Study
Intervention Model: Parallel Assignment
Masking: Double Blind (Subject, Investigator)
Primary Purpose: Treatment
Official Title: A Pilot Study of the Efficacy and Safety of BMS-512148 on Glycemic Control in Subjects With Type 2 Diabetes Treated Aggressively But Not Controlled on Combination Antihyperglycemic Therapy With Metformin and/or Thiazolidinedione (TZD) and Insulin.

Resource links provided by NLM:


Further study details as provided by Bristol-Myers Squibb:

Primary Outcome Measures:
  • Change from baseline in hemoglobin A1C [ Time Frame: at Week 12 ] [ Designated as safety issue: No ]

Secondary Outcome Measures:
  • Change from baseline in fasting plasma glucose [ Time Frame: at Week 12 ] [ Designated as safety issue: No ]
  • Change from baseline in the proportion of subjects achieving therapeutic glycemic responses [ Time Frame: at Week 12 ] [ Designated as safety issue: No ]
  • Change from baseline in the total daily dose of insulin [ Time Frame: at Week 12 ] [ Designated as safety issue: No ]

Enrollment: 67
Study Start Date: October 2006
Study Completion Date: March 2008
Primary Completion Date: March 2008 (Final data collection date for primary outcome measure)
Arms Assigned Interventions
Experimental: Cohort 1
20 mg
Drug: Dapagliflozin
Tablets, Oral, once daily, up to 12 weeks
Other Name: BMS-512148
Experimental: Cohort 2 - Arm 1
10 mg
Drug: Dapagliflozin
Tablets, Oral, once daily, up to 12 weeks
Other Name: BMS-512148
Experimental: Cohort 2 - Arm 2
20 mg
Drug: Dapagliflozin
Tablets, Oral, once daily, up to 12 weeks
Other Name: BMS-512148
Placebo Comparator: Cohort 2 - Arm 3 Drug: Placebo
Tablets, Oral, 0 mg, once daily, up to 12 weeks

  Eligibility

Ages Eligible for Study:   18 Years to 75 Years
Genders Eligible for Study:   Both
Accepts Healthy Volunteers:   No
Criteria

Inclusion Criteria:

  • Males and females, 18 to 75 years old, with type 2 diabetes with inadequate glycemic control
  • Subjects receiving insulin and metformin and/or a thiazolidinedione
  • Body Mass Index <=45.0 kg/m2
  • Serum creatinine <1.5 mg/dL for men or <1.4 mg/dL for women
  • No overt proteinuria (in subjects with a microalbumin/creatinine ratio ≥300 mg/g, the 24-hour urinary excretion of total protein must be <3 g/24 hrs)

Exclusion Criteria:

  • History of type 1 diabetes
  • AST and/or ALT >2.5 times the upper limit of normal
  • Creatinine kinase ≥3 times the upper limit of normal
  • Symptoms of severely uncontrolled diabetes
  • History of hypoglycemic unawareness
  • Currently unstable or serious cardiovascular, renal, hepatic, hematological, oncological, endocrine, psychiatric, or rheumatic diseases
  Contacts and Locations
Please refer to this study by its ClinicalTrials.gov identifier: NCT00357370

  Hide Study Locations
Locations
United States, Arkansas
Nea Clinic
Jonesboro, Arkansas, United States, 72401
United States, California
Valley Research
Fresno, California, United States, 93720
Bernstein, Richard
Greenbrae, California, United States, 94904
United States, Florida
Jacksonville Center For Clinical Research
Jacksonville, Florida, United States, 32205
United States, Georgia
Endocrine Research Solutions, Inc.
Roswell, Georgia, United States, 30076
United States, Indiana
Indiana University
Indianapolis, Indiana, United States, 46202
United States, Maryland
Model Clinical Research Llc
Baltimore, Maryland, United States, 21204
United States, Michigan
University Of Michigan
Ann Arbor, Michigan, United States, 48109
United States, Missouri
St. Louis Center For Clinical Research
St. Louis, Missouri, United States, 63128
United States, New York
Suny Upstate Medical University
Syracuse, New York, United States, 13210
United States, North Carolina
Mountain Diabetes And Endocrine Center
Asheville, North Carolina, United States, 28801
United States, Ohio
Your Diabetes Endocrine Nutrition Group
Mentor, Ohio, United States, 44060
United States, Texas
Research Institute Of Dallas, P.A.
Dallas, Texas, United States, 75231
Diabetes And Glandular Disease Research Associates, P.A.
San Antonio, Texas, United States, 78229
United States, Washington
Rainier Clinical Research Center
Renton, Washington, United States, 98055
United States, Wisconsin
Advanced Healthcare S.C.
Milwaukee, Wisconsin, United States, 53209
Canada, Manitoba
Local Institution
Winnipeg, Manitoba, Canada, R3E 3P4
Canada, New Brunswick
Local Institution
Bathurst, New Brunswick, Canada, E2A 4X7
Canada, Quebec
Local Institution
Gatineau, Quebec, Canada, J8V 2P5
Local Institution
Laval, Quebec, Canada, H7T 2P5
Local Institution
Longueuil, Quebec, Canada, J4N 1L6
Local Institution
Pointe-Claire, Quebec, Canada, H9R 4S3
Local Institution
Sherbrooke, Quebec, Canada, J1G 5K2
Sponsors and Collaborators
Bristol-Myers Squibb
Investigators
Study Director: Bristol-Myers Squibb Bristol-Myers Squibb
  More Information

Additional Information:
No publications provided

Responsible Party: Study Director, Bristol-Myers Squibb
ClinicalTrials.gov Identifier: NCT00357370     History of Changes
Other Study ID Numbers: MB102-009
Study First Received: July 26, 2006
Last Updated: September 10, 2010
Health Authority: United States: Food and Drug Administration

Additional relevant MeSH terms:
Diabetes Mellitus
Diabetes Mellitus, Type 2
Glucose Metabolism Disorders
Metabolic Diseases
Endocrine System Diseases
Hypoglycemic Agents
Physiological Effects of Drugs
Pharmacologic Actions

ClinicalTrials.gov processed this record on June 18, 2013